Compile Data Set for Download or QSAR
Found 71 of ic50 data for polymerid = 50004567
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50210162(CHEMBL3883534)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461172(CHEMBL4228518)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461178(CHEMBL4225777)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461174(CHEMBL4226676)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50112173(CHEMBL3608429)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50450868(CHEMBL4216679)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461179(CHEMBL4226151)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50029668(AZD-9291 | Osimertinib | US10085983, Compound AZD-...)copy SMILEScopy InChI
Affinity DataIC50: 2.10nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461175(CHEMBL4225565)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461176(CHEMBL4227084)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50450870(Mavelertinib | PF-06747775)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50437353(CHEMBL2408045)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human HER3 expressed in baculovirus/Sf21 system by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474F5DPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461180(CHEMBL4225306)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461177(CHEMBL4225951)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50461173(CHEMBL4226937)copy SMILEScopy InChI
Affinity DataIC50: 5.80nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) using poly (Glu, Tyr) as substrate after 40 mins by kinase-glo plus luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41V28PubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50112176(CHEMBL3608432)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467144(CHEMBL4288300)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467162(CHEMBL4282460)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50159360(CHEMBL3786098)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50611358(CHEMBL5285282)copy SMILES
Affinity DataIC50: 23nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467143(CHEMBL4283970)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467148(CHEMBL4294156)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50450867(CHEMBL4206501)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM149404(AVL-301 | CHEMBL3545308 | CNX-419 | CO-1686 | Roci...)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25X2CJZPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50611359(CHEMBL5282275)copy SMILES
Affinity DataIC50: 49nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467152(CHEMBL4283823)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467163(CHEMBL4290750)copy SMILEScopy InChI
Affinity DataIC50: 69nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467146(CHEMBL1379917)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467147(CHEMBL4283097)copy SMILEScopy InChI
Affinity DataIC50: 167nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467151(CHEMBL4293690)copy SMILEScopy InChI
Affinity DataIC50: 167nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467161(CHEMBL4278997)copy SMILEScopy InChI
Affinity DataIC50: 183nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467158(CHEMBL4280395)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467159(CHEMBL4288262)copy SMILEScopy InChI
Affinity DataIC50: 236nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467155(CHEMBL4276965)copy SMILEScopy InChI
Affinity DataIC50: 619nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467149(CHEMBL4287629)copy SMILEScopy InChI
Affinity DataIC50: 825nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467142(CHEMBL4293134)copy SMILEScopy InChI
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467153(CHEMBL4289682)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467164(CHEMBL4288761)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467166(CHEMBL4278031)copy SMILEScopy InChI
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467160(CHEMBL4281413)copy SMILEScopy InChI
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467157(CHEMBL4292110)copy SMILEScopy InChI
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467150(CHEMBL4284911)copy SMILEScopy InChI
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM494927((2S,4R)-1-((S)-2-(6-(4-(4-((4-((3-chloro-4-fluorop...)copy SMILEScopy InChI
Affinity DataIC50: 6.60E+3nMAssay Description:All compounds and PROTACs were serially diluted in three-fold increments using 100% DMSO, followed by an intermediate 10-fold dilution using Buffer A...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NS0Z1GUS Patent
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM494934(2-(2,6-dioxopiperidin-3-yl)-5-(2-(4-(2-((1-isoprop...)copy SMILEScopy InChI
Affinity DataIC50: 8.60E+3nMAssay Description:All compounds and PROTACs were serially diluted in three-fold increments using 100% DMSO, followed by an intermediate 10-fold dilution using Buffer A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NS0Z1GUS Patent
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467141(CHEMBL4283517)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467145(CHEMBL4282879)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467154(CHEMBL4286263)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467156(CHEMBL4286871)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
TargetReceptor tyrosine-protein kinase erbB-3(Homo sapiens (Human))
Wuxi AppTec

Curated by ChEMBL
LigandPNGBDBM50467165(CHEMBL4283061)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human GST-tagged EGFR L858R mutant cytoplasmic domain expressed in baculovirus expression system using FAM-labeled peptide ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SF2ZVSPubMed
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